99% Hormone Hormone Ipamorelin 2mg / Vial don Gina Jiki CAS 170851-70-4
CAS BA.: | 170851-70-4 | Tsarin kwayoyin halitta: | 38H49N9O5 |
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Kwayoyin Weight: | 711.853 | Gwaji: | 99.5% |
Bayyanar: | Farin Lyophilized Foda | Anfani: | Gyaran jiki |
Injectable peptide Hormone Ipamorelin 2mg / Vial don Gina Jiki CAS 170851-70-4
Saurin bayani
Sunan Samfur |
Ipamorelin
|
Laƙabi |
696: PN: WO2004005342 SHAFI: 46 da'awar sunadarai, Ipamorelin, NNC 26-0161
|
CAS |
170851-70-4
|
MF |
C38H49N9O5
|
MW |
711.853
|
Bayyanar |
Farin foda
|
Darasi |
Darajar Magunguna
|
Tsabta |
99%
|
Amfani |
Mai karɓar sinadarin ɓoye na haɓakar haɓakar G ne mai haɗarin furotin na G wanda yake ɗaure ghrelin kuma yana taka rawa a cikin homeostasis na makamashi da kuma daidaita nauyin jiki.
|
Bayani:
Ipamorelin wani sabon abu ne mai ban sha'awa wanda aka samu wanda yake samun kulawa sosai a cikin
gina jiki duniya. Yana da peptide na roba wanda ke da iko Ci gaban Hormon sake kayan. Kuma waɗannan abubuwan sakin GH sune abin sha'awa ga yan wasa da masu ginin jiki tunda zasu iya yin banbanci mai yawa a cikin adadin tsoka da zaka iya girma da kuma saurin saurin ƙona kitse.
Ipamorelin shine penta-peptide. (Aib-His-D-2-Nal-D- Phe-Lys-NH2) Kuma, ƙarfin da yake nunawa na iya zama daɗaɗa tsohuwar Ci Gaban Hormon (GH) ta tsufa. da gaske ana son sanin menene menene wannan peptide mai ban mamaki da zai iya yi, yaya ake amfani dashi, kuma yaya yake kwatankwacin sauran peptides na GHRP?
'Yan wasa suna shan Ipamorelin a cikin kwayar 200mcg -300mcg, sau biyu ko sau uku a kowace rana, ta amfani da karamin allurar insulin don yin allura.Yawancin lokaci sukan fara ne da karancin magani tunda illolin na iya hadawa da ciwon kai ko kuma abin da ake ji kamar kai-kawo. takenauke shi kowane lokaci amma ɗaukar shi kusan mintuna 30-45 kafin motsa jiki zai zama da kyau saboda bugun jini a cikin Girmancin Hormon (GH) wanda ya haifar da ƙimar girma.
Nazarin kan illar Ipamorelin akan ci gaban ƙashi, nauyin jiki, da sakin GH sun nuna wasu sakamako masu ban sha'awa. A cikin gwaji ɗaya, an gudanar da allurai iri-iri a cikin tsawon kwanaki 15 don gwada halayen ƙungiyar.
Akwai tasiri mai mahimmanci kuma mai dogaro akan haɓakar nauyin jiki duk da haka, ƙungiyar masu ba da magani ba ta nuna canji a cikin duka matakan IGF-I ba.Kuma rukunin maganin ba su samar da alamun jini na ƙashi ba
ci gaba. Misali, yawan kwayoyin halitta a cikin babban sashin tibia (shinbone) bai canza sosai ba. Wannan abu ne mai kyau saboda yana nuna ci gaban tsoka tare da rashin yiwuwar nakasar kashi ko guringuntsi.
Yanayin da pituitary yayi wa iVDose na Ipamorelin mai tsananin tashin hankali ya nuna cewa matakan GH plasma ya ragu musamman yayin da basu canza ba bayan kwatankwacin GHRH.Wannan a zahiri abu ne mai kyau kamar yadda yake nuna cewa Ipamorelin bazai iya rage samarwar GH na jikinka ba - kara nuna cewa Ipamorelin mai sake sakin GH ne.
Ipamorelin baya haifar da yunwa yana mai da fa'ida ga waɗanda ke cikin ƙuntataccen abincin kalori. Kuma a bayyane yake, tasirin tasirin Ipamorelin yana haɓaka idan aka haɗu tare da magungunan masu anabolic tunda su ma suna tasiri ga Growarfafa Hormon / Insulin Growth Factor saki da samarwa.
Bayanin IPamorelin
Bayani dalla-dalla
|
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Bayyanar |
Farin foda
|
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Bayyanar bayani |
Gaskiya
|
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Launi na bayani |
Launi mara launi
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PH |
tayin
|
||||||
Takamaiman Tsarin Gani (c = 0.5,95% HAc) |
tayin
|
||||||
Tsabta (na HPLC) |
98.00% ~ 99.90%
|
||||||
Jimlar Rashin Tsabta (ta HPLC) |
.002.00% ~ 0.05%
|
||||||
Rashin tsabta guda ɗaya (ta HPLC) |
.0.50% ~ 0.08%
|
||||||
Abun Ruwa (Karl Fischer) |
4.80%
|
||||||
Abun Cikin Acetate (na HPLC) |
6.80%
|
||||||
Abun Cikin Peptide (ta% N) |
88.00%
|
||||||
Amino Acaid Abun da ke ciki |
± 10% na ka'idoji
|
||||||
Assay (Ta hanyar anhydrous, acetic-free) |
95.0% ~ 105.0%
|
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Sauyawa
|
tayin |
Bayanan martaba:
Ipamorelin (ko NNC 26-0161) nasa ne na peptides na yau da kullun saboda GH ne ke sakin furotin; Sarkar ta gajere ce kuma kawai tana dauke ne da amino acid biyar. Yawan kwayar halitta / nauyinta shine 711.86 kuma tsarin kwayoyin shine C38H49N9O5. Ipamorelin an hada shi azaman sabon abu da kuma sabon abu na ghrelin saboda haka yana da ikon haɓaka motsin ciki. Akwai ƙananan gwaje-gwaje masu gudana na asibiti tare da ipamorelin a halin yanzu. Nazarin farko akan HGr-peptides gami da NNC 26-0161 an fara shi a farkon 1990s. Hakanan wannan mahaɗan bincike shine majami'ar zaɓaɓɓe ta G-hormone da agonist mai karɓar ghrelin. Kamar yadda sauran sunadaran ipamorelin sukeyi tare da masu karɓa na GHRP don sakin haɓakar girma daga gland. Amma sabanin 'yan sauran peptides na yanayin halittar wannan pentapeptide ba ya fitar da girman irin wannan mahadi kamar cortisol da acetylcholine, kuma wannan ya sa ya zama kyakkyawan ɗan takara don bincike na gaba. Bugu da ƙari, NNC 26-0161 ya fi daidaitaccen tsari na ghrelin kuma yana da tsawon rabin rai, kuma yana haifar da sakamako na biyu ta hanyar sanya jijiyoyi suyi farin ciki.
Aikace-aikace:
Ipamorelin shine peptide mai ban sha'awa wanda aka sha 300mcg sau biyu a kowace rana ko zaka iya rage maganin sau 3 a kowace rana, illolin sune saurin kai, Ina ba da shawarar a ɗauki wannan minti 30 kafin motsa jiki, tare da kaya, Ipamorelin sabon pentpeptide ne mai ƙarfi kuma mai ƙarfi. da takamaiman haɓakar haɓakar hormone (GH) - sakewa da kaddarorin. Tare da maƙasudin binciken sakamakon tasirin haɓakar ƙashi mai tsawo, nauyin jiki, da sakin GH, Ipamorelin a cikin allurai daban-daban (0, 18, 90 da 450 /g / day) an yi musu allura sau uku kowace rana don kwanaki 15 don gwada batutuwa,
Bayan lakabin Tetracycline na intravital a cikin ranakun 0, 6, da 13, an ƙaddara LGR ta hanyar auna tazara tsakanin maɗaukakiyar fitila a cikin tibia metaphysis kusa. Matsayi na Ipamorelin-ya haɓaka LGR daga 42 daym / rana a cikin ƙungiyar abin hawa zuwa 44, 50, da 52 μm / rana a cikin ƙungiyoyin kulawa. Hakanan akwai tasirin sakamako mai fa'ida akan ribar jikin. Maganin bai shafi duka matakan IGF-I ba, ko alamun magani na samuwar ƙashi da resorption ba.
Fuction:
Gina tsoka mai taushi, rage kitse a jiki da rage riƙe ruwa tare da Ipamorelin daga Cibiyar Kula da Matasa ta Har abada. Amfani don: Masu ginin jiki suna neman ƙara ƙarfi; Mutane na yau da kullun don asarar mai da ingancin haɓakar tsoka; Tsofaffi waɗanda ke neman fa'idodin tsufa; Saurin raunin rauni;
Amfani:
1. Kamfaninmu kwararren masana'antar samar da kayayyaki ne a kasar Sin a yankin magunguna na shekaru masu yawa. Yankunan isar da kayan mu: US, UK, Canada, Australia, Brazil, Russia, Portugal, Latvia, Switzerland, Iceland, Ukraine, Germany, France, Netherlands, Belgium, Peru, Sweden, New Zealand, Czech Republic, Lithuania, Ireland , Tunisia, Mexico, Girka, Puerto Rico, Thailand, Isra'ila da sauransu. Hanyar biyan kuɗi: T / T, unionungiyar yamma, Moneygram.
2. Hankali mai kunshin hankali.Kunshin hankali ya fi dacewa da ku za a zaɓa don ƙetare al'adu cikin aminci. Ko kuma idan kuna da kyakkyawar hanyarku, za a iya la'akari da shi.
3. Mafi inganci. Mai inganci mai kyau ne, da zarar an sami wata matsala, za a sake siyan kunshin
kai
4. Jirgin Tsaro: Ana jigilar kaya ta hanyar kar-ta-kwana (FedEx, UPS, DHL, EMS), ta hanyar iska. Za a ba da shawarar a tura muku kwararrun masu gabatarwa.
5. Muna da hannun jari, saboda haka zamu iya kaiwa da sauri a daidai lokacin da muka sami biyan.
6. Dumi bayan-sale sabis a gare ku 24/7. Duk wani tambayar ku za a warware ta ta farko da zarar ta samu
zai yiwu.
7. Za'a ba da ragi lokacin da kuka yi oda mai yawa.
Kayan Sayarwa Masu Zafi
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